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5m4h
From Proteopedia
(Difference between revisions)
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==Application of Off-Rate Screening in the Identification of Novel Pan-Isoform Inhibitors of Pyruvate Dehydrogenase Kinase== | ==Application of Off-Rate Screening in the Identification of Novel Pan-Isoform Inhibitors of Pyruvate Dehydrogenase Kinase== | ||
| - | <StructureSection load='5m4h' size='340' side='right' caption='[[5m4h]], [[Resolution|resolution]] 2.00Å' scene=''> | + | <StructureSection load='5m4h' size='340' side='right'caption='[[5m4h]], [[Resolution|resolution]] 2.00Å' scene=''> |
== Structural highlights == | == Structural highlights == | ||
<table><tr><td colspan='2'>[[5m4h]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Human Human]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=5M4H OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5M4H FirstGlance]. <br> | <table><tr><td colspan='2'>[[5m4h]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Human Human]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=5M4H OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=5M4H FirstGlance]. <br> | ||
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==See Also== | ==See Also== | ||
| - | *[[Heat Shock | + | *[[Heat Shock Protein structures|Heat Shock Protein structures]] |
== References == | == References == | ||
<references/> | <references/> | ||
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</StructureSection> | </StructureSection> | ||
[[Category: Human]] | [[Category: Human]] | ||
| + | [[Category: Large Structures]] | ||
[[Category: Baker, L M]] | [[Category: Baker, L M]] | ||
[[Category: Brough, P]] | [[Category: Brough, P]] | ||
Revision as of 07:17, 6 November 2019
Application of Off-Rate Screening in the Identification of Novel Pan-Isoform Inhibitors of Pyruvate Dehydrogenase Kinase
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Categories: Human | Large Structures | Baker, L M | Brough, P | Surgenor, A | Cancer | Fragment screening | Hsp90 | Kinase inhibitor | Off-rate screening | Pdhk | Pdk1 | Pdk2 | Pdk3 | Pdk4 | Signaling protein | Spr
