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6u09
From Proteopedia
(Difference between revisions)
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<StructureSection load='6u09' size='340' side='right'caption='[[6u09]], [[Resolution|resolution]] 1.79Å' scene=''> | <StructureSection load='6u09' size='340' side='right'caption='[[6u09]], [[Resolution|resolution]] 1.79Å' scene=''> | ||
== Structural highlights == | == Structural highlights == | ||
| - | <table><tr><td colspan='2'>[[6u09]] is a 4 chain structure. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=6U09 OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=6U09 FirstGlance]. <br> | + | <table><tr><td colspan='2'>[[6u09]] is a 4 chain structure with sequence from [http://en.wikipedia.org/wiki/Lk3_transgenic_mice Lk3 transgenic mice]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=6U09 OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=6U09 FirstGlance]. <br> |
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=EI9:3-{(1-oxo-1,2-dihydroisoquinolin-7-yl)[(pyridin-4-yl)methyl]sulfamoyl}benzene-1-sulfonyl+fluoride'>EI9</scene></td></tr> | </td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=EI9:3-{(1-oxo-1,2-dihydroisoquinolin-7-yl)[(pyridin-4-yl)methyl]sulfamoyl}benzene-1-sulfonyl+fluoride'>EI9</scene></td></tr> | ||
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[6u06|6u06]]</td></tr> | <tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[6u06|6u06]]</td></tr> | ||
| + | <tr id='gene'><td class="sblockLbl"><b>[[Gene|Gene:]]</b></td><td class="sblockDat">Eif4e ([http://www.ncbi.nlm.nih.gov/Taxonomy/Browser/wwwtax.cgi?mode=Info&srchmode=5&id=10090 LK3 transgenic mice])</td></tr> | ||
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=6u09 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=6u09 OCA], [http://pdbe.org/6u09 PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=6u09 RCSB], [http://www.ebi.ac.uk/pdbsum/6u09 PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=6u09 ProSAT]</span></td></tr> | <tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=6u09 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=6u09 OCA], [http://pdbe.org/6u09 PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=6u09 RCSB], [http://www.ebi.ac.uk/pdbsum/6u09 PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=6u09 ProSAT]</span></td></tr> | ||
</table> | </table> | ||
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</StructureSection> | </StructureSection> | ||
[[Category: Large Structures]] | [[Category: Large Structures]] | ||
| + | [[Category: Lk3 transgenic mice]] | ||
[[Category: Shoichet, B K]] | [[Category: Shoichet, B K]] | ||
[[Category: Taunton, J]] | [[Category: Taunton, J]] | ||
Revision as of 13:15, 18 December 2019
Discovery of Lysine-Targeted eIF4E Inhibitors through Covalent Docking
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