This old version of Proteopedia is provided for student assignments while the new version is undergoing repairs. Content and edits done in this old version of Proteopedia after March 1, 2026 will eventually be lost when it is retired in about June of 2026.


Apply for new accounts at the new Proteopedia. Your logins will work in both the old and new versions.


Peroxisome proliferator-activated receptor 3D structures

From Proteopedia

(Difference between revisions)
Jump to: navigation, search
Line 4: Line 4:
{{#tree:id=OrganizedByTopic|openlevels=0|
{{#tree:id=OrganizedByTopic|openlevels=0|
-
*'''PPARα'''
+
*'''PPARα''';Ligand-binding domain 201-468
-
**[[1k7l]] – hPPARα LBD + G2409544 + NCOA1 - human<br />
+
**[[1k7l]] – hPPARα + G2409544 + NCOA1 - human<br />
-
**[[3e94]] – hPPARα LBD + fatty acid activator <br />
+
**[[3e94]] – hPPARα + fatty acid activator <br />
-
**[[4bcr]], [[5hyk]] - hPPARα LBD + ligand<br />
+
**[[4bcr]], [[5hyk]] - hPPARα + ligand<br />
-
**[[1kkq]] – hPPARα LBD + GW6471 Antagonist + SMRT<br />
+
**[[1kkq]] – hPPARα + GW6471 Antagonist + SMRT<br />
-
**[[2npa]] - hPPARα LBD+ propanoic acid derivative + NCOA1<br />
+
**[[2npa]] - hPPARα + propanoic acid derivative + NCOA1<br />
-
**[[2p54]] - hPPARα LBD + NCOA1<br />
+
**[[2p54]] - hPPARα + NCOA1<br />
-
**[[2rew]] - hPPARα LBD + azetidinone derivative activator<br />
+
**[[2rew]] - hPPARα + azetidinone derivative activator<br />
-
**[[2znn]], [[2zno]], [[2znp]], [[2znq]], [[3kdu]], [[3vi8]], [[1i7g]], [[4bcr]], [[5hyk]] - hPPARα LBD+ agonist<br />
+
**[[2znn]], [[2zno]], [[2znp]], [[2znq]], [[3kdu]], [[3vi8]], [[1i7g]], [[4bcr]], [[5hyk]] - hPPARα + agonist<br />
-
**[[3fei]], [[3fej]], [[3g8i]], [[3sp6]] - hPPARα LBD+ agonist + NCOA1<br />
+
**[[3fei]], [[3fej]], [[3g8i]], [[3sp6]] - hPPARα + agonist + NCOA1<br />
-
**[[3et1]] - hPPARα LBD + NCOA1 + indole derivative
+
**[[3et1]] - hPPARα + NCOA1 + indole derivative
-
*'''PPARγ'''
+
*'''PPARγ''';Ligand-binding domain 202-475
-
**[[3prg]], [[2qmv]], [[1prg]] – hPPARγ LBD<br />
+
**[[3prg]], [[2qmv]], [[1prg]] – hPPARγ<br />
-
**[[6fzy]], [[6fzg]] - hPPARγ LBD (mutant) <br />
+
**[[6fzy]], [[6fzg]] - hPPARγ (mutant) <br />
-
**[[2zk0]], [[2zk1]], [[2zk2]], [[2zk3]], [[2zk4]], [[2zk5]], [[2zk6]], [[3vjh]], [[3vji]], [[4e4k]], [[4e4q]], [[4jl4]], [[5hzc]], [[4ci5]], [[4ci4]], [[6an1]], [[2f4b]], [[1zeo]], [[2ath]], [[2hwq]], [[2hwr]], [[2i4j]], [[2q59]], [[2q8s]], [[3b3k]], [[3bc5]], [[3cds]], [[3g9e]], [[3gbk]], [[3gz9]], [[3ia6]], [[3kdt]], [[3an3]], [[3an4]], [[3noa]], [[3r5n]], [[3r8a]], [[3vso]], [[3vsp]], [[2xkw]], [[3b0q]], [[3ho0]], [[3hod]], [[1knu]], [[1i7i]], [[1nyx]], [[2pob]], [[5azv]], [[6f2l]], [[6c5t]], [[6c5q]], [[5wr1]], [[5wr0]], [[5wqx]], [[6md2]], [[6md4]], [[6md1]], [[6md0]], [[6mcz]], [[6k0t]], [[6avi]], [[6aug]] – hPPARγ LBD + ligand <br />
+
**[[2zk0]], [[2zk1]], [[2zk2]], [[2zk3]], [[2zk4]], [[2zk5]], [[2zk6]], [[3vjh]], [[3vji]], [[4e4k]], [[4e4q]], [[4jl4]], [[5hzc]], [[4ci5]], [[4ci4]], [[6an1]], [[2f4b]], [[1zeo]], [[2ath]], [[2hwq]], [[2hwr]], [[2i4j]], [[2q59]], [[2q8s]], [[3b3k]], [[3bc5]], [[3cds]], [[3g9e]], [[3gbk]], [[3gz9]], [[3ia6]], [[3kdt]], [[3an3]], [[3an4]], [[3noa]], [[3r5n]], [[3r8a]], [[3vso]], [[3vsp]], [[2xkw]], [[3b0q]], [[3ho0]], [[3hod]], [[1knu]], [[1i7i]], [[1nyx]], [[2pob]], [[5azv]], [[6f2l]], [[6c5t]], [[6c5q]], [[5wr1]], [[5wr0]], [[5wqx]], [[6md2]], [[6md4]], [[6md1]], [[6md0]], [[6mcz]], [[6k0t]], [[6avi]], [[6aug]] – hPPARγ + ligand <br />
-
**[[4l98]], [[4l96]] - hPPARγ LBD (mutant) + ligand<br />
+
**[[4l98]], [[4l96]] - hPPARγ (mutant) + ligand<br />
-
**[[3r8i]] - hPPARγ LBD + ureidofibrate derivative<br />
+
**[[3r8i]] - hPPARγ + ureidofibrate derivative<br />
-
**[[6o67]], [[6o68]], [[6dgr]], [[6dgq]], [[6dgo]], [[6dgl]], [[6d8x]], [[6c1i]] - hPPARγ LBD + agonist<br />
+
**[[6o67]], [[6o68]], [[6dgr]], [[6dgq]], [[6dgo]], [[6dgl]], [[6d8x]], [[6c1i]] - hPPARγ + agonist<br />
-
**[[2g0h]], [[2g0g]], [[2i4p]], [[2i4z]], [[2q5g]], [[2q5p]], [[2q5s]], [[2q61]], [[2q6r]], [[3cdp]], [[3d6d]], [[4em9]], [[4ema]], [[4prg]], [[2q6s]], [[5f9b]], [[4yt1]], [[3wmh]], [[6d3e]] - hPPARγ LBD+ partial agonist<br />
+
**[[2g0h]], [[2g0g]], [[2i4p]], [[2i4z]], [[2q5g]], [[2q5p]], [[2q5s]], [[2q61]], [[2q6r]], [[3cdp]], [[3d6d]], [[4em9]], [[4ema]], [[4prg]], [[2q6s]], [[5f9b]], [[4yt1]], [[3wmh]], [[6d3e]] - hPPARγ + partial agonist<br />
-
**[[2om9]] - hPPARγ LBD + cannabinoid<br />
+
**[[2om9]] - hPPARγ + cannabinoid<br />
-
**[[3b0r]], [[5lsg]], [[4r6s]], [[4r2u]], [[4r06]], [[6dh9]], [[6dcu]], [[6dbh]] - hPPARγ LBD + antagonist<br />
+
**[[3b0r]], [[5lsg]], [[4r6s]], [[4r2u]], [[4r06]], [[6dh9]], [[6dcu]], [[6dbh]] - hPPARγ + antagonist<br />
-
**[[3osi]], [[3osw]], [[3pba]] - hPPARγ LBD + bisphenol derivative<br />
+
**[[3osi]], [[3osw]], [[3pba]] - hPPARγ + bisphenol derivative<br />
-
**[[2p4y]], [[3adt]], [[3adu]], [[3adw]], [[3et3]], [[2hfp]], [[3ty0]] - hPPARγ LBD + modulator<br />
+
**[[2p4y]], [[3adt]], [[3adu]], [[3adw]], [[3et3]], [[2hfp]], [[3ty0]] - hPPARγ + modulator<br />
-
**[[2zvt]] - hPPARγ LBD (mutant) + modulator<br />
+
**[[2zvt]] - hPPARγ (mutant) + modulator<br />
-
**[[2vsr]], [[2vst]], [[2vv0]], [[2vv1]], [[2vv2]], [[2vv3]], [[2vv4]], [[3x1i]], [[3x1h]], [[3wj5]], [[3wj4]], [[3po9]], [[3sz1]] - hPPARγ LBD + fatty acid activator<br />
+
**[[2vsr]], [[2vst]], [[2vv0]], [[2vv1]], [[2vv2]], [[2vv3]], [[2vv4]], [[3x1i]], [[3x1h]], [[3wj5]], [[3wj4]], [[3po9]], [[3sz1]] - hPPARγ + fatty acid activator<br />
-
**[[3ads]], [[3adx]], [[5u5l]], [[4xum]], [[4xuh]], [[4xta]], [[4xld]], [[6d5a]] - hPPARγ LBD + anti-inflammatory drug<br />
+
**[[3ads]], [[3adx]], [[5u5l]], [[4xum]], [[4xuh]], [[4xta]], [[4xld]], [[6d5a]] - hPPARγ + anti-inflammatory drug<br />
-
**[[4oj4]] - hPPARγ LBD (mutant) + anti-inflammatory drug<br />
+
**[[4oj4]] - hPPARγ (mutant) + anti-inflammatory drug<br />
-
**[[3adv]] - hPPARγ LBD + serotonin<br />
+
**[[3adv]] - hPPARγ + serotonin<br />
-
**[[3k8s]], [[3et0]], [[2yfe]], [[4a4v]], [[4a4w]], [[4jaz]], [[5tto]], [[4pwl]], [[4pvu]], [[5y2t]], [[5y2o]], [[5ugm]], [[6dha]] - hPPARγ LBD + antidiabetic drug<br />
+
**[[3k8s]], [[3et0]], [[2yfe]], [[4a4v]], [[4a4w]], [[4jaz]], [[5tto]], [[4pwl]], [[4pvu]], [[5y2t]], [[5y2o]], [[5ugm]], [[6dha]] - hPPARγ + antidiabetic drug<br />
-
**[[4o8f]] - hPPARγ LBD (mutant) + antidiabetic drug<br />
+
**[[4o8f]] - hPPARγ (mutant) + antidiabetic drug<br />
-
**[[6enq]] - hPPARγ LBD + antifibrotic drug<br />
+
**[[6enq]] - hPPARγ + antifibrotic drug<br />
*PPARγ complex with polypeptide
*PPARγ complex with polypeptide
-
**[[1wm0]] – hPPARγ LBD+ NCAO2 peptide + agonist<br />
+
**[[1wm0]] – hPPARγ + NCAO2 peptide + agonist<br />
-
**[[5dwl]], [[5dvc]], [[5dv8]], [[5dv6]], [[5dv3]], [[5dsh]] - hPPARγ LBD+ NCOA2 peptide + inhibitor<br />
+
**[[5dwl]], [[5dvc]], [[5dv8]], [[5dv6]], [[5dv3]], [[5dsh]] - hPPARγ + NCOA2 peptide + inhibitor<br />
-
**[[1zgy]] – hPPARγ LBD+ antidiabetic drug + nuclear receptor peptide<br />
+
**[[1zgy]] – hPPARγ + antidiabetic drug + nuclear receptor peptide<br />
-
**[[2gtk]], [[3qt0]], [[5gtp]], [[5gto]], [[5gtn]], [[6jq7]], [[6izm]], [[6ilq]], [[6ijs]], [[6ijr]], [[6icj]], [[5ycp]], [[5ycn]] - hPPARγ LBD+ NCOA1 peptide<br />
+
**[[2gtk]], [[3qt0]], [[5gtp]], [[5gto]], [[5gtn]], [[6jq7]], [[6izm]], [[6ilq]], [[6ijs]], [[6ijr]], [[6icj]], [[5ycp]], [[5ycn]] - hPPARγ + NCOA1 peptide<br />
-
**[[3cs8]], [[3u9q]]- hPPARγ LBD + PGC-1A peptide<br />
+
**[[3cs8]], [[3u9q]]- hPPARγ + PGC-1A peptide<br />
-
**[[3cwd]] - hPPARγ LBD + NCOA1-2 peptide<br />
+
**[[3cwd]] - hPPARγ + NCOA1-2 peptide<br />
-
**[[5two]], [[6izn]], [[6fzp]], [[6fzj]], [[6fzf]] - hPPARγ LBD + modulating ligand<br />
+
**[[5two]], [[6izn]], [[6fzp]], [[6fzj]], [[6fzf]] - hPPARγ + modulating ligand<br />
-
**[[3fur]], [[3kmg]], [[3v9t]], [[3v9v]], [[3v9y]], [[4f9m]], [[3b1m]], [[3lmp]] - hPPARγ LBD + SRC-1 peptide + modulator<br />
+
**[[3fur]], [[3kmg]], [[3v9t]], [[3v9v]], [[3v9y]], [[4f9m]], [[3b1m]], [[3lmp]] - hPPARγ + SRC-1 peptide + modulator<br />
-
**[[4fgy]], [[2prg]] - hPPARγ LBD + antidiabetic agent + NCOA1 peptide<br />
+
**[[4fgy]], [[2prg]] - hPPARγ + antidiabetic agent + NCOA1 peptide<br />
-
**[[6ad9]] - hPPARγ LBD + anticancer agent + NCOA1 peptide<br />
+
**[[6ad9]] - hPPARγ + anticancer agent + NCOA1 peptide<br />
-
**[[3s9s]], [[3t03]], [[2fvj]]- hPPARγ LBD + NCOA1 peptide + partial agonist<br />
+
**[[3s9s]], [[3t03]], [[2fvj]]- hPPARγ + NCOA1 peptide + partial agonist<br />
-
**[[4y29]], [[2fvj]], [[5azt]] - hPPARγ LBD + NCOA1 peptide + ligand<br />
+
**[[4y29]], [[2fvj]], [[5azt]] - hPPARγ + NCOA1 peptide + ligand<br />
-
**[[3h0a]] - hPPARγ LBD + SRC 1 + retinoic acid receptor α + retinoic acid + partial agonist<br />
+
**[[3h0a]] - hPPARγ + SRC 1 + retinoic acid receptor α + retinoic acid + partial agonist<br />
-
**[[1k74]], [[1rdt]], [[1fm9]] - hPPARγ LBD + NCOA1 + retinoic acid receptor α + retinoic acid + agonist<br />
+
**[[1k74]], [[1rdt]], [[1fm9]] - hPPARγ + NCOA1 + retinoic acid receptor α + retinoic acid + agonist<br />
-
**[[5ji0]] - hPPARγ LBD + retinoic acid receptor + NCOA1 peptide + antidiabetic drug <br />
+
**[[5ji0]] - hPPARγ + retinoic acid receptor + NCOA1 peptide + antidiabetic drug <br />
-
**[[3dzu]], [[3e00]], [[3dzy]] - hPPARγ LBD + DNA + retinoic acid receptor α + NCOA2 peptide + retinoic acid<br />
+
**[[3dzu]], [[3e00]], [[3dzy]] - hPPARγ + DNA + retinoic acid receptor α + NCOA2 peptide + retinoic acid<br />
-
**[[1fm6]] - hPPARγ LBD + antidiabetic drug + retinoic acid receptor α + NCOA2 peptide + retinoic acid<br />
+
**[[1fm6]] - hPPARγ + antidiabetic drug + retinoic acid receptor α + NCOA2 peptide + retinoic acid<br />
-
**[[3vn2]], [[4hee]], [[4prg]] - hPPARγ LBD + NCOA1 peptide + activator<br />
+
**[[3vn2]], [[4hee]], [[4prg]] - hPPARγ + NCOA1 peptide + activator<br />
-
**[[6ms7]] - hPPARγ LBD + PGC1 LXXLL<br />
+
**[[6ms7]] - hPPARγ + PGC1 LXXLL<br />
-
**[[6dgp]], [[5z6s]], [[5z5s]] - hPPARγ LBD + coactivator peptide<br />
+
**[[6dgp]], [[5z6s]], [[5z5s]] - hPPARγ + coactivator peptide<br />
-
**[[6d94]] - hPPARγ LBD + mediator of RNA polymerase II peptide<br />
+
**[[6d94]] - hPPARγ + mediator of RNA polymerase II peptide<br />
-
*'''PPARδ'''
+
*'''PPARδ''';Ligand-binding domain 171-441
-
**[[2gwx]] – hPPARδ LBD<br />
+
**[[2gwx]] – hPPARδ<br />
-
**[[2env]] – hPPARδ zinc finger domain<br />
+
**[[2env]] – hPPARδ zinc finger domain 72-146 - NMR<br />
**[[2baw]], [[2b50]], [[2awh]] – hPPARδ + Vaccenic Acid<br />
**[[2baw]], [[2b50]], [[2awh]] – hPPARδ + Vaccenic Acid<br />
-
**[[3gwx]] – hPPARδ LBD + 5,8,11,14,17-Eicosapentaenoic Acid<br />
+
**[[3gwx]] – hPPARδ + 5,8,11,14,17-Eicosapentaenoic Acid<br />
-
**[[3dy6]] – hPPARδ LBD + anthranilic acid <br />
+
**[[3dy6]] – hPPARδ + anthranilic acid <br />
**[[3et2]], [[1gwx]] – hPPARδ + fatty acid<br />
**[[3et2]], [[1gwx]] – hPPARδ + fatty acid<br />
-
**[[2j14]], [[2xyj]], [[2xyw]], [[2xyx]], [[3oz0]], [[3sp9]], [[5u3q]], [[5u3r]], [[5u3s]], [[5u3t]], [[5u3u]], [[5u3v]], [[5u3w]], [[5u3x]], [[5u3y]], [[5u3z]], [[5u40]], [[5u41]], [[5u42]], [[5u43]], [[5u44]], [[5u45]], [[1gwx]], [[3tkm]], [[1y0s]], [[5u46]], [[5y7x]] - hPPARδ LBD + agonist<br />
+
**[[2j14]], [[2xyj]], [[2xyw]], [[2xyx]], [[3oz0]], [[3sp9]], [[5u3q]], [[5u3r]], [[5u3s]], [[5u3t]], [[5u3u]], [[5u3v]], [[5u3w]], [[5u3x]], [[5u3y]], [[5u3z]], [[5u40]], [[5u41]], [[5u42]], [[5u43]], [[5u44]], [[5u45]], [[1gwx]], [[3tkm]], [[1y0s]], [[5u46]], [[5y7x]] - hPPARδ + agonist<br />
-
**[[3peq]] - hPPARδ LBD + partial agonist<br />
+
**[[3peq]] - hPPARδ + partial agonist<br />
-
**[[3d5f]] - hPPARδ LBD + phenoxy derivative<br />
+
**[[3d5f]] - hPPARδ + phenoxy derivative<br />
-
**[[5xmx]], [[6a6p]], [[5zxi]] - hPPARδ LBD + inhibitor<br />
+
**[[5xmx]], [[6a6p]], [[5zxi]] - hPPARδ + inhibitor<br />
}}
}}
[[Category:Topic Page]]
[[Category:Topic Page]]

Revision as of 08:52, 21 September 2020

3D Structures of PPAR

Updated on 21-September-2020

Proteopedia Page Contributors and Editors (what is this?)

Michal Harel, Jaime Prilusky

Personal tools