This old version of Proteopedia is provided for student assignments while the new version is undergoing repairs. Content and edits done in this old version of Proteopedia after March 1, 2026 will eventually be lost when it is retired in about June of 2026.


Apply for new accounts at the new Proteopedia. Your logins will work in both the old and new versions.


4nqn

From Proteopedia

(Difference between revisions)
Jump to: navigation, search
Line 1: Line 1:
==Crystal Structure of the bromodomain of human BRD9 in complex with a triazolo-phthalazine ligand==
==Crystal Structure of the bromodomain of human BRD9 in complex with a triazolo-phthalazine ligand==
-
<StructureSection load='4nqn' size='340' side='right' caption='[[4nqn]], [[Resolution|resolution]] 1.73&Aring;' scene=''>
+
<StructureSection load='4nqn' size='340' side='right'caption='[[4nqn]], [[Resolution|resolution]] 1.73&Aring;' scene=''>
== Structural highlights ==
== Structural highlights ==
-
<table><tr><td colspan='2'>[[4nqn]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Human Human]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4NQN OCA]. For a <b>guided tour on the structure components</b> use [http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4NQN FirstGlance]. <br>
+
<table><tr><td colspan='2'>[[4nqn]] is a 1 chain structure with sequence from [https://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=4NQN OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=4NQN FirstGlance]. <br>
-
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat"><scene name='pdbligand=Y1Z:2-CHLORO-N-[5-(3-METHYL[1,2,4]TRIAZOLO[3,4-A]PHTHALAZIN-6-YL)-2-(MORPHOLIN-4-YL)PHENYL]BENZENESULFONAMIDE'>Y1Z</scene></td></tr>
+
</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=Y1Z:2-CHLORO-N-[5-(3-METHYL[1,2,4]TRIAZOLO[3,4-A]PHTHALAZIN-6-YL)-2-(MORPHOLIN-4-YL)PHENYL]BENZENESULFONAMIDE'>Y1Z</scene></td></tr>
-
<tr id='related'><td class="sblockLbl"><b>[[Related_structure|Related:]]</b></td><td class="sblockDat">[[4nqm|4nqm]]</td></tr>
+
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=4nqn FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4nqn OCA], [https://pdbe.org/4nqn PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=4nqn RCSB], [https://www.ebi.ac.uk/pdbsum/4nqn PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=4nqn ProSAT]</span></td></tr>
-
<tr id='gene'><td class="sblockLbl"><b>[[Gene|Gene:]]</b></td><td class="sblockDat">BRD9 ([http://www.ncbi.nlm.nih.gov/Taxonomy/Browser/wwwtax.cgi?mode=Info&srchmode=5&id=9606 HUMAN])</td></tr>
+
-
<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[http://oca.weizmann.ac.il/oca-docs/fgij/fg.htm?mol=4nqn FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=4nqn OCA], [http://pdbe.org/4nqn PDBe], [http://www.rcsb.org/pdb/explore.do?structureId=4nqn RCSB], [http://www.ebi.ac.uk/pdbsum/4nqn PDBsum], [http://prosat.h-its.org/prosat/prosatexe?pdbcode=4nqn ProSAT]</span></td></tr>
+
</table>
</table>
 +
== Function ==
 +
[https://www.uniprot.org/uniprot/BRD9_HUMAN BRD9_HUMAN] May play a role in chromatin remodeling and regulation of transcription.
==See Also==
==See Also==
-
*[[Bromodomain-containing protein|Bromodomain-containing protein]]
+
*[[Bromodomain-containing protein 3D structures|Bromodomain-containing protein 3D structures]]
__TOC__
__TOC__
</StructureSection>
</StructureSection>
-
[[Category: Human]]
+
[[Category: Homo sapiens]]
-
[[Category: Arrowsmith, C H]]
+
[[Category: Large Structures]]
-
[[Category: Bountra, C]]
+
[[Category: Arrowsmith CH]]
-
[[Category: Delft, F von]]
+
[[Category: Bountra C]]
-
[[Category: Edwards, A M]]
+
[[Category: Edwards AM]]
-
[[Category: Fedorov, O]]
+
[[Category: Fedorov O]]
-
[[Category: Felletar, I]]
+
[[Category: Felletar I]]
-
[[Category: Filippakopoulos, P]]
+
[[Category: Filippakopoulos P]]
-
[[Category: Knapp, S]]
+
[[Category: Knapp S]]
-
[[Category: Martin, S]]
+
[[Category: Martin S]]
-
[[Category: Picaud, S]]
+
[[Category: Picaud S]]
-
[[Category: Structural genomic]]
+
[[Category: Von Delft F]]
-
[[Category: Bromodomain]]
+
-
[[Category: Inhibition]]
+
-
[[Category: Sgc]]
+
-
[[Category: Small molecule inhibitor]]
+
-
[[Category: Transcription]]
+
-
[[Category: Transcription-inhibitor complex]]
+

Revision as of 08:42, 11 January 2023

Crystal Structure of the bromodomain of human BRD9 in complex with a triazolo-phthalazine ligand

PDB ID 4nqn

Drag the structure with the mouse to rotate

Proteopedia Page Contributors and Editors (what is this?)

OCA

Personal tools