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7zy6

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'''Unreleased structure'''
 
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The entry 7zy6 is ON HOLD until Paper Publication
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==Identification of M4205 a highly selective inhibitor of cKIT mutations for unresectable metastatic or recurrent GIST==
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<StructureSection load='7zy6' size='340' side='right'caption='[[7zy6]], [[Resolution|resolution]] 3.09&Aring;' scene=''>
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Authors: Graedler, U., Lammens, A.
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== Structural highlights ==
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<table><tr><td colspan='2'>[[7zy6]] is a 1 chain structure with sequence from [https://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=7ZY6 OCA]. For a <b>guided tour on the structure components</b> use [https://proteopedia.org/fgij/fg.htm?mol=7ZY6 FirstGlance]. <br>
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Description: Identification of M4205 a highly selective inhibitor of cKIT mutations for unresectable metastatic or recurrent GIST
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</td></tr><tr id='ligand'><td class="sblockLbl"><b>[[Ligand|Ligands:]]</b></td><td class="sblockDat" id="ligandDat"><scene name='pdbligand=KCI:5-imidazo[1,2-a]pyridin-3-yl-~{N}-[(1~{R})-1-(6-pyrrolidin-1-ylpyridin-3-yl)ethyl]pyridin-3-amine'>KCI</scene></td></tr>
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[[Category: Unreleased Structures]]
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<tr id='resources'><td class="sblockLbl"><b>Resources:</b></td><td class="sblockDat"><span class='plainlinks'>[https://proteopedia.org/fgij/fg.htm?mol=7zy6 FirstGlance], [http://oca.weizmann.ac.il/oca-bin/ocaids?id=7zy6 OCA], [https://pdbe.org/7zy6 PDBe], [https://www.rcsb.org/pdb/explore.do?structureId=7zy6 RCSB], [https://www.ebi.ac.uk/pdbsum/7zy6 PDBsum], [https://prosat.h-its.org/prosat/prosatexe?pdbcode=7zy6 ProSAT]</span></td></tr>
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[[Category: Graedler, U]]
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</table>
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[[Category: Lammens, A]]
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__TOC__
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</StructureSection>
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[[Category: Homo sapiens]]
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[[Category: Large Structures]]
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[[Category: Graedler U]]
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[[Category: Lammens A]]

Revision as of 12:38, 22 February 2023

Identification of M4205 a highly selective inhibitor of cKIT mutations for unresectable metastatic or recurrent GIST

PDB ID 7zy6

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