3byz
From Proteopedia
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{{STRUCTURE_3byz| PDB=3byz | SCENE= }} | {{STRUCTURE_3byz| PDB=3byz | SCENE= }} | ||
- | + | ===2-Amino-1,3-thiazol-4(5H)-ones as Potent and Selective 11-Hydroxysteroid Dehydrogenase Type 1 Inhibitors=== | |
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+ | The line below this paragraph, {{ABSTRACT_PUBMED_18419108}}, adds the Publication Abstract to the page | ||
+ | (as it appears on PubMed at http://www.pubmed.gov), where 18419108 is the PubMed ID number. | ||
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+ | {{ABSTRACT_PUBMED_18419108}} | ||
==About this Structure== | ==About this Structure== | ||
3BYZ is a [[Single protein]] structure of sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=3BYZ OCA]. | 3BYZ is a [[Single protein]] structure of sequence from [http://en.wikipedia.org/wiki/Homo_sapiens Homo sapiens]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=3BYZ OCA]. | ||
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+ | ==Reference== | ||
+ | 2-amino-1,3-thiazol-4(5H)-ones as potent and selective 11beta-hydroxysteroid dehydrogenase type 1 inhibitors: enzyme-ligand co-crystal structure and demonstration of pharmacodynamic effects in C57Bl/6 mice., Johansson L, Fotsch C, Bartberger MD, Castro VM, Chen M, Emery M, Gustafsson S, Hale C, Hickman D, Homan E, Jordan SR, Komorowski R, Li A, McRae K, Moniz G, Matsumoto G, Orihuela C, Palm G, Veniant M, Wang M, Williams M, Zhang J, J Med Chem. 2008 May 22;51(10):2933-43. Epub 2008 Apr 18. PMID:[http://www.ncbi.nlm.nih.gov/pubmed/18419108 18419108] | ||
[[Category: 11-beta-hydroxysteroid dehydrogenase]] | [[Category: 11-beta-hydroxysteroid dehydrogenase]] | ||
[[Category: Homo sapiens]] | [[Category: Homo sapiens]] | ||
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[[Category: Steroid metabolism]] | [[Category: Steroid metabolism]] | ||
[[Category: Transmembrane]] | [[Category: Transmembrane]] | ||
- | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on | + | |
+ | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Wed Jul 2 22:04:10 2008'' |
Revision as of 19:04, 2 July 2008
2-Amino-1,3-thiazol-4(5H)-ones as Potent and Selective 11-Hydroxysteroid Dehydrogenase Type 1 Inhibitors
Template:ABSTRACT PUBMED 18419108
About this Structure
3BYZ is a Single protein structure of sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
2-amino-1,3-thiazol-4(5H)-ones as potent and selective 11beta-hydroxysteroid dehydrogenase type 1 inhibitors: enzyme-ligand co-crystal structure and demonstration of pharmacodynamic effects in C57Bl/6 mice., Johansson L, Fotsch C, Bartberger MD, Castro VM, Chen M, Emery M, Gustafsson S, Hale C, Hickman D, Homan E, Jordan SR, Komorowski R, Li A, McRae K, Moniz G, Matsumoto G, Orihuela C, Palm G, Veniant M, Wang M, Williams M, Zhang J, J Med Chem. 2008 May 22;51(10):2933-43. Epub 2008 Apr 18. PMID:18419108
Page seeded by OCA on Wed Jul 2 22:04:10 2008
Categories: 11-beta-hydroxysteroid dehydrogenase | Homo sapiens | Single protein | Jordan, S R. | Li, V. | Zhang, J. | Alpha beta | Endoplasmic reticulum | Glycoprotein | Lipid metabolism | Membrane | Microsome | Nadp | Oxidoreductase | Polymorphism | Rossmann fold | Signal-anchor | Steroid metabolism | Transmembrane