3d4n
From Proteopedia
Line 1: | Line 1: | ||
{{Seed}} | {{Seed}} | ||
- | [[Image:3d4n. | + | [[Image:3d4n.png|left|200px]] |
<!-- | <!-- | ||
Line 46: | Line 46: | ||
[[Category: Transmembrane]] | [[Category: Transmembrane]] | ||
- | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on | + | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Tue Jul 29 16:18:36 2008'' |
Revision as of 13:18, 29 July 2008
Crystal Structure of Human 11-beta-Hydroxysteroid Dehydrogenase (HSD1) in Complex with Sulfonamide Inhibitor
Template:ABSTRACT PUBMED 18553955
About this Structure
3D4N is a Single protein structure of sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
Discovery of Novel, Potent Benzamide Inhibitors of 11beta-Hydroxysteroid Dehydrogenase Type 1 (11beta-HSD1) Exhibiting Oral Activity in an Enzyme Inhibition ex Vivo Model., Julian LD, Wang Z, Bostick T, Caille S, Choi R, Degraffenreid M, Di Y, He X, Hungate RW, Jaen JC, Liu J, Monshouwer M, McMinn D, Rew Y, Sudom A, Sun D, Tu H, Ursu S, Walker N, Yan X, Ye Q, Powers JP, J Med Chem. 2008 Jun 14;. PMID:18553955
Page seeded by OCA on Tue Jul 29 16:18:36 2008
Categories: 11-beta-hydroxysteroid dehydrogenase | Homo sapiens | Single protein | Liu, J. | Sudom, A. | Walker, N P. | Wang, Z. | 11beta | Dehydrogenase | Endoplasmic reticulum | Glycoprotein | Hydroxysteroid | Lipid metabolism | Membrane | Microsome | Nadp | Oxidoreductase | Polymorphism | Signal-anchor | Steroid metabolism | Transmembrane