3eqr
From Proteopedia
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[[Category: Homo sapiens]] | [[Category: Homo sapiens]] | ||
[[Category: Non-specific protein-tyrosine kinase]] | [[Category: Non-specific protein-tyrosine kinase]] | ||
- | [[Category: | + | [[Category: Liu, J.]] |
+ | [[Category: Walker, N P.C.]] | ||
+ | [[Category: Wang, Z.]] | ||
[[Category: Ack1]] | [[Category: Ack1]] | ||
[[Category: Alternative splicing]] | [[Category: Alternative splicing]] | ||
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[[Category: Tyrosine-protein kinase]] | [[Category: Tyrosine-protein kinase]] | ||
- | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on | + | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Wed Dec 10 15:41:52 2008'' |
Revision as of 13:41, 10 December 2008
Crystal Structure of Ack1 with compound T74
Template:ABSTRACT PUBMED 18993068
About this Structure
3EQR is a 2 chains structure of sequences from Homo sapiens. Full crystallographic information is available from OCA.
Reference
Identification and optimization of N3,N6-diaryl-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamines as a novel class of ACK1 inhibitors., Kopecky DJ, Hao X, Chen Y, Fu J, Jiao X, Jaen JC, Cardozo MG, Liu J, Wang Z, Walker NP, Wesche H, Li S, Farrelly E, Xiao SH, Kayser F, Bioorg Med Chem Lett. 2008 Dec 15;18(24):6352-6. Epub 2008 Nov 1. PMID:18993068
Page seeded by OCA on Wed Dec 10 15:41:52 2008
Categories: Homo sapiens | Non-specific protein-tyrosine kinase | Liu, J. | Walker, N P.C. | Wang, Z. | Ack1 | Alternative splicing | Atp-binding | Cell membrane | Kinase | Magnesium | Membrane | Metal-binding | Nucleotide-binding | Phosphoprotein | Polymorphism | Sh3 domain | Transferase | Tyrosine-protein kinase