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3uza
From Proteopedia
Thermostabilised Adenosine A2A receptor in complex with 6-(2,6-Dimethylpyridin-4-yl)-5-phenyl-1,2,4-triazin-3-amine
Template:ABSTRACT PUBMED 22220592
About this Structure
3uza is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Congreve M, Andrews SP, Dore AS, Hollenstein K, Hurrell E, Langmead CJ, Mason JS, Ng IW, Tehan B, Zhukov A, Weir M, Marshall FH. Discovery of 1,2,4-Triazine Derivatives as Adenosine A(2A) Antagonists using Structure Based Drug Design. J Med Chem. 2012 Mar 8;55(5):1898-903. Epub 2012 Jan 27. PMID:22220592 doi:10.1021/jm201376w
Categories: Homo sapiens | Andrews, S P. | Congreve, M. | Dore, A S. | Hollenstein, K. | Hurrell, E. | Langmead, C J. | Marshall, F H. | Mason, J S. | Ng, I W. | Tehan, B. | Weir, M. | Zhukov, A. | 7tm | G-protein | Gpcr | Membrane protein | Signaling protein
