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4an3
From Proteopedia
Crystal structures of human MEK1 with carboxamide-based allosteric inhibitor XL518 (GDC-0973), or related analogs.
About this Structure
4an3 is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Categories: Homo sapiens | Mitogen-activated protein kinase kinase | Aay, N. | Anand, N K. | Blazey, C M. | Bowles, O J. | Bussenius, J. | Costanzo, S. | Curtis, J K. | Defina, S C. | Dubenko, L. | Engst, S. | Johnston, S. | Joshi, A A. | Kennedy, A R. | Kim, A I. | Koltun, E S. | Lougheed, J C. | Manalo, J C.L. | Martini, J F. | Nuss, J M. | Peto, C J. | Rice, K D. | Tsang, T H. | Yu, P. | Allosteric inhibition | Atp-binding | Map2k1 | Transferase
