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5aau
From Proteopedia
Unreleased structure
The entry 5aau is ON HOLD until Paper Publication
Authors: Norman, R.A., Bradbury, R.H., de Almeida, C., Andrews, D.M., Ballard, P., Buttar, D., Callis, R.J., Currie, G.S., Curwen, J.O., Davies, C.D., de Savi, C., Donald, C.S., Feron, L.J.L., Glossop, S.C., Hayter, B.R., Karoutchi, G., Lamont, S.G., MacFaul, P., Moss, T., Pearson, S.E., Rabow, A.A., Tonge, M., Walker, G.E., Weir, H.M., Wilson, Z.
Description: Optimization of a novel binding motif to to (E)-3-(3,5-difluoro-4-(( 1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-2,3,4,9-tetrahydro-1H-pyrido(3,4-b)indol-1-yl)phenyl)acrylic acid (AZD9496), a potent and orally bioavailable selective estrogen receptor downregulator and antagonist
Categories: Unreleased Structures | Walker, G.E | Rabow, A.A | Wilson, Z | Curwen, J.O | Moss, T | Karoutchi, G | Ballard, P | Glossop, S.C | Davies, C.D | De Almeida, C | Buttar, D | Donald, C.S | Andrews, D.M | De Savi, C | Callis, R.J | Hayter, B.R | Macfaul, P | Feron, L.J.L | Norman, R.A | Weir, H.M | Tonge, M | Lamont, S.G | Pearson, S.E | Currie, G.S | Bradbury, R.H
