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1c5o
From Proteopedia
Contents |
STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR
Template:ABSTRACT PUBMED 10779411
About this Structure
1c5o is a 3 chain structure of Hirudin and Thrombin with sequence from Hirudo medicinalis and Homo sapiens. Full crystallographic information is available from OCA.
See Also
Reference
- Katz BA, Mackman R, Luong C, Radika K, Martelli A, Sprengeler PA, Wang J, Chan H, Wong L. Structural basis for selectivity of a small molecule, S1-binding, submicromolar inhibitor of urokinase-type plasminogen activator. Chem Biol. 2000 Apr;7(4):299-312. PMID:10779411
Categories: Hirudo medicinalis | Homo sapiens | Thrombin | Chan, H. | Katz, B A. | Luong, C. | Mackman, R. | Martelli, A. | Radika, K. | Sprengeler, P A. | Wang, J. | Wong, L. | Blood clotting-hydrolase inhibitor complex | S1 site inhibitor | Selective | Structure-based drug design | Trypsin | Urokinase
