2vts
From Proteopedia
IDENTIFICATION OF N-(4-PIPERIDINYL)-4-(2,6-DICHLOROBENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXAMIDE (AT7519), A NOVEL CYCLIN DEPENDENT KINASE INHIBITOR USING FRAGMENT-BASED X-RAY CRYSTALLOGRAPHY AND STRUCTURE BASED DRUG DESIGN.
About this Structure
2VTS is a 1 chain structure of sequence from Homo sapiens. Full crystallographic information is available from OCA.
Page seeded by OCA on Mon Feb 16 15:09:52 2009
Categories: Homo sapiens | Berdini, V. | Boulstridge, J A. | Brien, M A.O. | Carr, M G. | Cross, D M. | Danillon, D. | Davis, D J. | Devine, L A. | Early, T R. | Feltell, R E. | Lewis, E J. | Mcmenamin, R L. | Navarro, E F. | Reilly, M O. | Reule, M. | Saxty, G. | Seavers, L C.A. | Smith, D M. | Squires, M S. | Trewartha, G. | Walker, M T. | Woodhead, A J. | Woolford, A J.A. | Wyatt, P G. | Atp-binding | Cell cycle | Cell division | Fragment screening | Kinase | Mitosis | Nucleotide-binding | Phosphoprotein | Phosphorylation | Polymorphism | Protein kinase | Serine/threonine protein kinase | Serine/threonine-protein kinase | Structure based drug design | Transferase