3ezr
From Proteopedia
Contents |
CDK-2 with indazole inhibitor 17 bound at its active site
Template:ABSTRACT PUBMED 19097791
About this Structure
3ezr is a 1 chain structure of Cell Division Protein Kinase 2 with sequence from Homo sapiens. Full crystallographic information is available from OCA.
See Also
Reference
- Trujillo JI, Kiefer JR, Huang W, Thorarensen A, Xing L, Caspers NL, Day JE, Mathis KJ, Kretzmer KK, Reitz BA, Weinberg RA, Stegeman RA, Wrightstone A, Christine L, Compton R, Li X. 2-(6-Phenyl-1H-indazol-3-yl)-1H-benzo[d]imidazoles: design and synthesis of a potent and isoform selective PKC-zeta inhibitor. Bioorg Med Chem Lett. 2009 Feb 1;19(3):908-11. Epub 2008 Dec 6. PMID:19097791 doi:10.1016/j.bmcl.2008.11.105
Categories: Cyclin-dependent kinase | Homo sapiens | Caspers, N L. | Christine, L. | Compton, R. | Day, J E. | Huang, W. | Kiefer, J R. | Kretzmer, K K. | Li, X. | Mathis, K J. | Reitz, B A. | Stegeman, R A. | Thorarensen, A. | Trujillo, J I. | Weinberg, R A. | Wrightstone, A. | Xing, L. | Atp-binding | Cell cycle | Cell division | Inhibitor | Kinase | Mitosis | Nucleotide-binding | Phosphoprotein | Pkc | Protein kinase | Serine/threonine-protein kinase | Transferase