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3en6
From Proteopedia
Targeted polypharmacology: crystal structure of the c-Src kinase domain in complex with PP102, a multitargeted kinase inhibitor
Template:ABSTRACT PUBMED 18849971
About this Structure
3EN6 is a 2 chains structure of sequences from Gallus gallus. Full crystallographic information is available from OCA.
Reference
- Apsel B, Blair JA, Gonzalez B, Nazif TM, Feldman ME, Aizenstein B, Hoffman R, Williams RL, Shokat KM, Knight ZA. Targeted polypharmacology: discovery of dual inhibitors of tyrosine and phosphoinositide kinases. Nat Chem Biol. 2008 Nov;4(11):691-9. Epub 2008 Oct 12. PMID:18849971 doi:http://dx.doi.org/10.1038/nchembio.117
Page seeded by OCA on Tue Feb 17 21:57:17 2009
Categories: Gallus gallus | Non-specific protein-tyrosine kinase | Apsel, B. | Blair, J A. | Knight, Z A. | Shokat, K M. | Alternative splicing | Atp-binding | Inhibitor | Kinase | Kinase-inhibitor complex | Lipoprotein | Multitarget | Myristate | Nucleotide-binding | Phosphoinositide | Phosphoprotein | Polypharmacology | Proto-oncogene | Pyrazolopyrimidine | Sh2 domain | Sh3 domain | Signaling | Src | Transferase | Tyrosine | Tyrosine-protein kinase
