This old version of Proteopedia is provided for student assignments while the new version is undergoing repairs. Content and edits done in this old version of Proteopedia after March 1, 2026 will eventually be lost when it is retired in about June of 2026.
Apply for new accounts at the new Proteopedia. Your logins will work in both the old and new versions.
3udd
From Proteopedia
Tankyrase-1 in complex with small molecule inhibitor
Template:ABSTRACT PUBMED 22260203
About this Structure
3udd is a 2 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Shultz MD, Kirby CA, Stams T, Chin DN, Blank J, Charlat O, Cheng H, Cheung AK, Feng Y, Fortin PD, Hood T, Tyagi V, Xu M, Zhang B, Shao W. [1,2,4]Triazol-3-ylsulfanylmethyl)-3-phenyl-[1,2,4]oxadiazoles: Antagonists of the Wnt pathway that inhibit tankyrase 1&2 via novel adenosine pocket binding. J Med Chem. 2012 Jan 19. PMID:22260203 doi:10.1021/jm2011222
