3o95

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Template:STRUCTURE 3o95

Contents 1 Crystal Structure of Human DPP4 Bound to TAK-100 2 About this Structure 3 See Also 4 Reference

Crystal Structure of Human DPP4 Bound to TAK-100

Template:ABSTRACT PUBMED 21218817

About this Structure

3o95 is a 4 chain structure of Dipeptidyl peptidase with sequence from Homo sapiens. Full crystallographic information is available from OCA.

See Also

• Dipeptidyl peptidase

Reference

• Miyamoto Y, Banno Y, Yamashita T, Fujimoto T, Oi S, Moritoh Y, Asakawa T, Kataoka O, Yashiro H, Takeuchi K, Suzuki N, Ikedo K, Kosaka T, Tsubotani S, Tani A, Sasaki M, Funami M, Amano M, Yamamoto Y, Aertgeerts K, Yano J, Maezaki H. Discovery of a 3-Pyridylacetic Acid Derivative (TAK-100) as a Potent, Selective and Orally Active Dipeptidyl Peptidase IV (DPP-4) Inhibitor. J Med Chem. 2011 Jan 10. PMID:21218817 doi:10.1021/jm101236h