3kmc

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Template:STRUCTURE 3kmc

Contents 1 Crystal structure of catalytic domain of TACE with tartrate-based inhibitor 2 About this Structure 3 See Also 4 Reference

Crystal structure of catalytic domain of TACE with tartrate-based inhibitor

Template:ABSTRACT PUBMED 20022498

About this Structure

3kmc is a 2 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.

See Also

• A Disintegrin And Metalloproteinase

Reference

• Rosner KE, Guo Z, Orth P, Shipps GW Jr, Belanger DB, Chan TY, Curran PJ, Dai C, Deng Y, Girijavallabhan VM, Hong L, Lavey BJ, Lee JF, Li D, Liu Z, Popovici-Muller J, Ting PC, Vaccaro H, Wang L, Wang T, Yu W, Zhou G, Niu X, Sun J, Kozlowski JA, Lundell DJ, Madison V, McKittrick B, Piwinski JJ, Shih NY, Arshad Siddiqui M, Strickland CO. The discovery of novel tartrate-based TNF-alpha converting enzyme (TACE) inhibitors. Bioorg Med Chem Lett. 2010 Feb 1;20(3):1189-93. Epub 2009 Dec 5. PMID:20022498 doi:10.1016/j.bmcl.2009.12.004