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4ly9
From Proteopedia
Human GKRP complexed to AMG-1694 [(2R)-1,1,1-trifluoro-2-{4-[(2S)-2-{[(3S)-3-methylmorpholin-4-yl]methyl}-4-(thiophen-2-ylsulfonyl)piperazin-1-yl]phenyl}propan-2-ol] and sorbitol-6-phosphate
Function
[GCKR_HUMAN] Inhibits glucokinase by forming an inactive complex with this enzyme.
About this Structure
4ly9 is a 2 chain structure. Full crystallographic information is available from OCA.
