2bmc
From Proteopedia
AURORA-2 T287D T288D COMPLEXED WITH PHA-680632
Template:ABSTRACT PUBMED 15828847
About this Structure
2bmc is a 6 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Fancelli D, Berta D, Bindi S, Cameron A, Cappella P, Carpinelli P, Catana C, Forte B, Giordano P, Giorgini ML, Mantegani S, Marsiglio A, Meroni M, Moll J, Pittala V, Roletto F, Severino D, Soncini C, Storici P, Tonani R, Varasi M, Vulpetti A, Vianello P. Potent and selective Aurora inhibitors identified by the expansion of a novel scaffold for protein kinase inhibition. J Med Chem. 2005 Apr 21;48(8):3080-4. PMID:15828847 doi:http://dx.doi.org/10.1021/jm049076m
Categories: Homo sapiens | Non-specific serine/threonine protein kinase | Berta, D. | Bindi, S. | Cameron, A D. | Catana, C. | Fancelli, D. | Forte, B. | Giordano, P. | Izzo, G. | Mantegani, S. | Meroni, M. | Moll, J. | Pittala, V. | Rusconi, L. | Sagliano, A. | Severino, D. | Storici, P. | Tonani, R. | Varasi, M. | Vianello, P. | Vulpetti, A. | Atp-binding | Cell cycle | Phosphorylation | Serine/threonine-protein kinase | Transferase