4bqg
From Proteopedia
structure of HSP90 with an inhibitor bound
Template:ABSTRACT PUBMED 24100158
About this Structure
4bqg is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Brasca MG, Mantegani S, Amboldi N, Bindi S, Caronni D, Casale E, Ceccarelli W, Colombo N, De Ponti A, Donati D, Ermoli A, Fachin G, Felder ER, Ferguson RD, Fiorelli C, Guanci M, Isacchi A, Pesenti E, Polucci P, Riceputi L, Sola F, Visco C, Zuccotto F, Fogliatto G. Discovery of NMS-E973 as novel, selective and potent inhibitor of heat shock protein 90 (Hsp90). Bioorg Med Chem. 2013 Nov 15;21(22):7047-63. doi: 10.1016/j.bmc.2013.09.018. Epub, 2013 Sep 19. PMID:24100158 doi:http://dx.doi.org/10.1016/j.bmc.2013.09.018
Categories: Homo sapiens | Amboldi, N. | Bindi, S. | Brasca, M G. | Caronni, D. | Casale, E. | Ceccarelli, W. | Colombo, N. | DePonti, A. | Donati, D. | Ermoli, A. | Fachin, G. | Felder, E R. | Ferguson, R D. | Fiorelli, C. | Fogliatto, G. | Guanci, M. | Isacchi, A. | Mantegani, S. | Pesenti, E. | Polucci, P. | Riceputi, L. | Sola, F. | Visco, C. | Zuccotto, F. | Chaperone
