3d3e
From Proteopedia
Crystal Structure of Human 11-beta-Hydroxysteroid Dehydrogenase (HSD1) in Complex with Benzamide Inhibitor
Template:ABSTRACT PUBMED 18553955
About this Structure
3D3E is a Single protein structure of sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
Discovery of Novel, Potent Benzamide Inhibitors of 11beta-Hydroxysteroid Dehydrogenase Type 1 (11beta-HSD1) Exhibiting Oral Activity in an Enzyme Inhibition ex Vivo Model., Julian LD, Wang Z, Bostick T, Caille S, Choi R, Degraffenreid M, Di Y, He X, Hungate RW, Jaen JC, Liu J, Monshouwer M, McMinn D, Rew Y, Sudom A, Sun D, Tu H, Ursu S, Walker N, Yan X, Ye Q, Powers JP, J Med Chem. 2008 Jun 14;. PMID:18553955
Page seeded by OCA on Thu Jul 3 11:32:56 2008
Categories: 11-beta-hydroxysteroid dehydrogenase | Homo sapiens | Single protein | Liu, J. | Sudom, A. | Walker, N P. | Wang, Z. | 11beta | Dehydrogenase | Endoplasmic reticulum | Glycoprotein | Hydroxysteroid | Lipid metabolism | Membrane | Microsome | Nadp | Oxidoreductase | Polymorphism | Signal-anchor | Steroid metabolism | Transmembrane