3czr
From Proteopedia
Crystal Structure of Human 11-beta-Hydroxysteroid Dehydrogenase (HSD1) in Complex with Arylsulfonylpiperazine Inhibitor
Template:ABSTRACT PUBMED 18511278
About this Structure
3CZR is a Single protein structure of sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
Discovery and initial SAR of arylsulfonylpiperazine inhibitors of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-HSD1)., Sun D, Wang Z, Di Y, Jaen JC, Labelle M, Ma J, Miao S, Sudom A, Tang L, Tomooka CS, Tu H, Ursu S, Walker N, Yan X, Ye Q, Powers JP, Bioorg Med Chem Lett. 2008 Jun 15;18(12):3513-6. Epub 2008 May 10. PMID:18511278
Page seeded by OCA on Sun Jul 27 17:53:08 2008
Categories: 11-beta-hydroxysteroid dehydrogenase | Homo sapiens | Single protein | Sudom, A. | Walker, N P. | Wang, Z. | 11beta | Dehydrogenase | Endoplasmic reticulum | Glycoprotein | Hydroxysteroid | Lipid metabolism | Membrane | Microsome | Nadp | Oxidoreductase | Polymorphism | Signal-anchor | Steroid metabolism | Transmembrane