2r9s

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Template:STRUCTURE 2r9s

c-Jun N-terminal Kinase 3 with 3,5-Disubstituted Quinoline inhibitor

Template:ABSTRACT PUBMED 17911023

About this Structure

2R9S is a 2 chains structure with sequences from Homo sapiens. Full crystallographic information is available from OCA.

Reference

  • Jiang R, Duckett D, Chen W, Habel J, Ling YY, LoGrasso P, Kamenecka TM. 3,5-Disubstituted quinolines as novel c-Jun N-terminal kinase inhibitors. Bioorg Med Chem Lett. 2007 Nov 15;17(22):6378-82. Epub 2007 Aug 26. PMID:17911023 doi:S0960-894X(07)01011-6

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