3qrk
From Proteopedia
The crystal structure of human abl1 kinase domain in complex with DP-987
Template:ABSTRACT PUBMED 21481795
About this Structure
3qrk is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Chan WW, Wise SC, Kaufman MD, Ahn YM, Ensinger CL, Haack T, Hood MM, Jones J, Lord JW, Lu WP, Miller D, Patt WC, Smith BD, Petillo PA, Rutkoski TJ, Telikepalli H, Vogeti L, Yao T, Chun L, Clark R, Evangelista P, Gavrilescu LC, Lazarides K, Zaleskas VM, Stewart LJ, Van Etten RA, Flynn DL. Conformational control inhibition of the BCR-ABL1 tyrosine kinase, including the gatekeeper T315I mutant, by the switch-control inhibitor DCC-2036. Cancer Cell. 2011 Apr 12;19(4):556-68. PMID:21481795 doi:10.1016/j.ccr.2011.03.003
Categories: Homo sapiens | Non-specific protein-tyrosine kinase | Ahn, Y M. | Chan, W W. | Chun, L. | Clark, R. | Ensinger, C L. | Etten, R A.Van. | Evangelista, P. | Flynn, D L. | Gavrilescu, L C. | Haack, T. | Hood, M M. | Jones, J. | Kaufman, M D. | Lazarides, K. | Lord, J W. | Lu, W P. | Miller, D. | Patt, W C. | Petillo, P A. | Rutkoski, T J. | Smith, B D. | Stewart, L J. | Telikepalli, H. | Vogeti, L. | Wise, S C. | Yao, T. | Zaleskas, V M.