3p79

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Template:STRUCTURE 3p79

P38 inhibitor-bound

Template:ABSTRACT PUBMED 22014550

About this Structure

3p79 is a 1 chain structure with sequence from Mus musculus. Full crystallographic information is available from OCA.

Reference

  • Moffett K, Konteatis Z, Nguyen D, Shetty R, Ludington J, Fujimoto T, Lee KJ, Chai X, Namboodiri H, Karpusas M, Dorsey B, Guarnieri F, Bukhtiyarova M, Springman E, Michelotti E. Discovery of a novel class of non-ATP site DFG-out state p38 inhibitors utilizing computationally assisted virtual fragment-based drug design (vFBDD). Bioorg Med Chem Lett. 2011 Sep 28. PMID:22014550 doi:10.1016/j.bmcl.2011.09.078

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