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3sdg
From Proteopedia
Ethionamide Boosters Part 2: Combining Bioisosteric Replacement and Structure-Based Drug Design to Solve Pharmacokinetic Issues in a Series of Potent 1,2,4-Oxadiazole EthR Inhibitors.
Template:ABSTRACT PUBMED 22098589
About this Structure
3sdg is a 1 chain structure with sequence from Mycobacterium tuberculosis. Full crystallographic information is available from OCA.
Reference
- Flipo M, Desroses M, Lecat-Guillet N, Villemagne B, Blondiaux N, Leroux F, Piveteau C, Mathys V, Flament MP, Siepmann J, Villeret V, Wohlkonig A, Wintjens R, Soror SH, Christophe T, Jeon HK, Locht C, Brodin P, Deprez BP, Baulard A, Willand N. Ethionamide Boosters Part 2: Combining Bioisosteric Replacement and Structure-Based Drug Design to Solve Pharmacokinetic Issues in a Series of Potent 1,2,4-Oxadiazole EthR Inhibitors. J Med Chem. 2011 Nov 20. PMID:22098589 doi:10.1021/jm200825u
Categories: Mycobacterium tuberculosis | Baulard, A R. | Blondiaux, N. | Brodin, P. | Christophe, T. | Desroses, M. | Flament, M P. | Flipo, M. | Jeon, H K. | Lecat-Guillet, N. | Leroux, F. | Locht, C. | Mathys, V. | Piveteau, C. | Siepmann, J. | Soror, S H. | Villemagne, B. | Villeret, V. | Willand, N | Wintjens, R. | Wohlkonig, A. | Prez, BD. | Dna | Dna binding | Dna binding protein | Inhibitor | Tetr-family | Transcription repressor-inhibitor complex | Transcritptional regulatory repressor
