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4d9t
From Proteopedia
Rsk2 C-terminal Kinase Domain with inhibitor (E)-methyl 3-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrolo[2,3-d]pyrimidin-6-yl)-2-cyanoacrylate
Template:ABSTRACT PUBMED 22466421
About this Structure
4d9t is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Serafimova IM, Pufall MA, Krishnan S, Duda K, Cohen MS, Maglathlin RL, McFarland JM, Miller RM, Frodin M, Taunton J. Reversible targeting of noncatalytic cysteines with chemically tuned electrophiles. Nat Chem Biol. 2012 Apr 1;8(5):471-6. doi: 10.1038/nchembio.925. PMID:22466421 doi:10.1038/nchembio.925
Categories: Homo sapiens | Non-specific serine/threonine protein kinase | Cohen, M S. | Duda, K. | Frodin, M. | Krishnan, S. | Maglathlin, R L. | McFarland, J M. | Miller, R M. | Pufall, M A. | Serafimova, I M. | Taunton, J. | Inhibitor | Kinase | Migration | Phosphorylation | Reversible | Thiol | Transferase-transferase inhibitor complex
