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4app
From Proteopedia
Crystal Structure of the Human p21-Activated Kinase 4 in Complex with (S)-N-(5-(3-benzyl-1-methylpiperazine-4-carbonyl)-6,6-dimethyl-1,4,5, 6-tetrahydropyrrolo(3,4-c)pyrazol-3-yl)-3-phenoxybenzamide
Template:ABSTRACT PUBMED 22554206
About this Structure
4app is a 1 chain structure with sequence from Homo sapiens. Full crystallographic information is available from OCA.
Reference
- Guo C, McAlpine I, Zhang J, Knighton DD, Kephart S, Johnson MC, Li H, Bouzida D, Yang A, Dong L, Marakovits J, Tikhe J, Richardson P, Guo LC, Kania R, Edwards MP, Kraynov E, Christensen J, Piraino J, Lee J, Dagostino E, Del-Carmen C, Deng YL, Smeal T, Murray BW. Discovery of Pyrroloaminopyrazoles as Novel PAK Inhibitors. J Med Chem. 2012 May 24;55(10):4728-39. Epub 2012 May 14. PMID:22554206 doi:10.1021/jm300204j
Categories: Homo sapiens | Non-specific serine/threonine protein kinase | Bouzida, D. | Christensen, J. | Dagostino, E. | Del-Carmen, C. | Deng, Y L. | Dong, L. | Edwards, M P. | Guo, C. | Guo, L C. | Johnson, M C. | Kania, R. | Kephart, S. | Knighton, D D. | Kraynov, E. | Lee, J. | Li, H. | Marakovits, J. | Mcalpine, I. | Murray, B W. | Piraino, J. | Richardson, P. | Smeal, T. | Tikhe, J. | Wang, C. | Yang, A. | Zhang, J. | Protein kinase | Transferase
