Fibroblast growth factor receptor 3D receptor
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3D structures of fibroblast growth factor receptor
Updated on 03-July-2025
FGFR1
8jqi
– hFGFR1 + PLC gamma – human – Cryo EM
FGFR1 tyrosine kinase domain (TKD) residues 458-765
4uwy
– hFGFR1 TKD
1fgk
,
3kxx
,
3ky2
,
4rwi
,
5flf
– hFGFR1 TKD (mutant)
4wun
,
5am6
,
5ew8
,
5o49
,
5o4a
,
6c1o
,
6mzq
,
6mzw
,
8xlo
,
8xlq
,
8xz7
,
8y22
,
9cd5
– hFGFR1 TKD + inhibitor
1agw
,
1fgi
,
2fgi
,
3c4f
,
3js2
,
3rhx
,
4f63
,
4f64
,
4f65
,
3tt0
,
4nk9
,
4nka
,
4nks
,
5b7v
,
5am7
,
4rwj
,
4rwk
,
4rwl
,
4uwb
,
4uwc
,
4zsa
,
5uq0
,
5vnd
,
5ur1
,
6c18
,
6c19
,
6c1b
,
6c1c
,
5z0s
,
6agx
,
6itj
,
6nvl
,
6p68
,
6p69
,
7ozb
,
7ozd
,
7ozf
,
7ozy
,
7wct
,
7wcw
,
7wcx
– hFGFR1 TKD (mutant) + inhibitor
8yki
– hFGFR1 TKD + anti-cancer drug
5zv2
,
7wcl
,
8jmz
– hFGFR1 TKD (mutant) + anti-cancer drug
3krj
– hFGFR1 TKD residues 538-678, 753-922 (mutant) + inhibitor
1xr0
– hFGFR1 residues 409-430 + FGFR signaling adaptor N terminal - NMR
3gqi
– hFGFR1 TKD (mutant) with PTR + ACP
3gql
– hFGFR1 TKD (mutant) + substrate
FGFR1 ligand-binding domain (LBD) D1 residues 35-208
2cr3
– hFGFR1 LBD D1 - NMR
2ckn
– FGFR1 LBD D1 – mouse - NMR
FGFR1 LBD D1 complex with FGF
5w59
– hFGFR1 LBD D1 + FGF9
FGFR1 LBD D2,D3 residues 142-365 complex with FGF
3ojv
– hFGFR1 LBD D2,D3 (mutant) + hFGF1 - human
1cvs
– hFGFR1 LBD D2,D3 (mutant) + hFGF2 (mutant)
1evt
– hFGFR1 LBD D2,D3 + hFGF1
1fq9
– hFGFR1 (mutant) LBD D2,D3 + hFGF2 (mutant) + HS
5w21
.
7ysh
– hFGFR1 LBD D2,D3 + hFGF23 + klotho
FGFR2
FGFR2 tyrosine kinase domain 413-821
1gjo
,
1oec
,
2psq
– hFGFR2 TKD
2pvy
,
2pwl
,
2py3
,
2pz5
,
2pzp
,
2pzr
,
2q0b
,
4j95
,
4j96
,
4j97
,
4j98
,
4j99
,
5ugx
,
5uhn
,
5ui0
– hFGFR2 TKD (mutant) + ACP
5ugl
– hFGFR2 TKD (mutant) + ANP
3b2t
– hFGFR2 TKD (mutant) + adenosine derivative
2pvf
– hFGFR2 TKD with PTR + ACP + substrate peptide
3cly
,
6v6q
– hFGFR2 TKD (mutant) with PTR + ACP
5eg3
– hFGFR2 TKD (mutant) with PTR + ACP + phospholipase C γ
3ri1
,
6lvk
,
6lvl
,
8e1x
,
8h75
,
8stg
,
8u1f
,
8w2x
,
8w38
,
8w3d
– hFGFR2 TKD + inhibitor
7kia
,
7kie
,
8swe
,
9u3n
– hFGFR2 TKD (mutant) + inhibitor
FGFR2 ligand-binding domain 134-249
3dar
,
3caf
,
3euu
– hFGFR2 LBD D2 150-249
8om6
– hFGFR2 LBD D2 (mutant)
1wvz
– hFGFR2 LBD D2 - NMR
4wv1
– hFGFR2 LBD D2 + antibody
6l4o
– hFGFR2 LBD D2 (mutant) + API5
4hwu
– hFGFR2 LBD D1 45-127
FGFR2 complex with FGF
1e0o
– hFGFR2 (mutant) LBD D2,D3 + hFGF1 (mutant) + HS
3oj2
,
3ojm
– hFGFR2 (mutant) LBD D2,D3 + hFGF1
1djs
– hFGFR2 LBD D2,D3 (mutant) + hFGF1
1ev2
,
1ii4
,
1iil
– hFGFR2 LBD D2,D3 + hFGF2 (mutant)
4j23
– hFGFR2 LBD D2,D3 (mutant) + hFGF2 (mutant) + inhibitor
3cu1
– hFGFR2 LBD D2 + hFGF1
2fdb
– hFGFR2 LBD D2,D3 + hFGF8b
1nun
– hFGFR2 LBD D2,D3 + hFGF10
FGFR3
3grw
– hFGFR3 LBD D2,D3 + antibody
2lzl
– hFGFR3 residues 357-399 – NMR
4k33
– hFGFR3 TKD (mutant)
6lvm
,
7dhl
,
8udt
,
8udu
,
8udv
,
9cd7
,
9d1x
– hFGFR3 TKD + inhibitor
6pnx
– hFGFR3 TKD (mutant) + ACP
FGFR3 complex with FGF
1ry7
– hFGFR3 LBD + hFGF1
7ysu
– hFGFR3 LBD D2,D3 + hFGF23 + klotho – Cryo EM
FGFR4
FGFR4 tyrosine kinase domain
4tye
,
4tyg
,
4tyi
,
4tyj
– hFGFR4 TKD
4qqj
,
4qqt
– hFGFR4 TKD (mutant)
5jkg
,
5nwz
,
5nud
,
6nvg
,
6nvh
,
6nvi
,
6nvj
,
6nvk
,
6v9c
,
7dtz
,
7f3m
,
7v29
,
7vjl
,
7wct
,
7ybo
,
7yc1
,
7yc3
,
8w5c
– hFGFR4 TKD + inhibitor
7tyd
– hFGFR4 TKD + protein inhibitor
6yi8
– hFGFR4 TKD + drug
5xff
,
5xfj
,
6iuo
,
6iup
,
6jpe
,
6jpj
,
7v29
,
7wcw
,
7wcx
,
7ybp
,
7ybx
,
8kh6
,
8kh7
,
8kh8
,
8kh9
– hFGFR4 TKD (mutant) + inhibitor
4qrc
,
4r6v
,
4qqc
,
4qq5
,
4uxq
,
4xcu
– hFGFR4 TKD (mutant) + irreversible inhibitor
FGFR4 LBD
6j6y
– hFGFR4 LBD D2 + antibody
7n1j
,
7tyd
– hFGFR4 LBD D3 + binder
Proteopedia Page Contributors and Editors
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Michal Harel
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