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Article title matches

1. Category:Phosphodiesterase 10a pde10a pde inhibitor (73 bytes)
   1: ...t of pages with the keyword Phosphodiesterase 10a pde10a pde inhibitor
2. Category:Pde10a (37 bytes)
   1: List of pages with the keyword Pde10a
3. Category:Pde10a inhibitor (47 bytes)
   1: List of pages with the keyword Pde10a inhibitor

Page text matches

1. 4hf4 (3,232 bytes)
   2: ==Crystal Structure of PDE10A with a biaryl ether inhibitor (1-(1-(3-(4-(benzo[...
   14: ... novel binding modes to the catalytic site of the PDE10A enzyme.
   16: Discovery of selective biaryl ethers as PDE10A inhibitors: Improvement in potency and mitigation...
2. 2oup (2,784 bytes)
   2: ==crystal structure of PDE10A==
3. 4bbx (3,962 bytes)
   2: ...iscovery of a potent, selective and orally active PDE10A inhibitor for the treatment of schizophrenia==
   14: ...hibitor of PDE10A with high striatal occupancy of PDE10A, promising in vivo efficacy in different rodent b...
   16: ...iscovery of a potent, selective and orally active PDE10A inhibitor for the potential treatment of schizoph...
4. 2ovv (3,981 bytes)
   24: ...otent and selective brain penetrable inhibitor of PDE10A.
   26: ...a series of 6,7-dimethoxy-4-pyrrolidylquinazoline PDE10A inhibitors.,Chappie TA, Humphrey JM, Allen MP, Es...
5. 2zmf (6,026 bytes)
   8: ..."><b>[[Gene|Gene:]]</b></td><td class="sblockDat">PDE10A ([https://www.ncbi.nlm.nih.gov/Taxonomy/Browser/w...
   26: ...he adenine base is specifically recognized by the PDE10A GAF-B domain in a unique manner, through residues...
6. 4heu (3,180 bytes)
   2: ==Crystal Structure of PDE10A with a biaryl ether inhibitor ((1-(3-(4-((1H-benz...
   14: ... novel binding modes to the catalytic site of the PDE10A enzyme.
   16: Discovery of selective biaryl ethers as PDE10A inhibitors: Improvement in potency and mitigation...
7. 2wey (4,759 bytes)
   24: .... Using crystals of human phosphodiesterase 10a (hPDE10a) as an example of such a challenging crystallogra...
   26: ...igand crystal complexes, exemplified by the human PDE10a-papaverine structure.,Andersen OA, Schonfeld DL, ...
8. 3hqw (4,342 bytes)
   2: ==Discovery of novel inhibitors of PDE10A==
   24: ...3-yl)-phenoxymethyl]-quinoline (PF-2545920). This PDE10A inhibitor is the first reported clinical entry fo...
   26: ... Schizophrenia (dagger) dagger Coordinates of the PDE10A crystal structures have been deposited in the Pro...
9. 3hqy (4,410 bytes)
   2: ==Discovery of novel inhibitors of PDE10A==
   24: ...3-yl)-phenoxymethyl]-quinoline (PF-2545920). This PDE10A inhibitor is the first reported clinical entry fo...
   26: ... Schizophrenia (dagger) dagger Coordinates of the PDE10A crystal structures have been deposited in the Pro...
10. 3hqz (4,404 bytes)
    2: ==Discovery of novel inhibitors of PDE10A==
    24: ...3-yl)-phenoxymethyl]-quinoline (PF-2545920). This PDE10A inhibitor is the first reported clinical entry fo...
    26: ... Schizophrenia (dagger) dagger Coordinates of the PDE10A crystal structures have been deposited in the Pro...
11. 3hr1 (4,414 bytes)
    2: ==Discovery of novel inhibitors of PDE10A==
    24: ...3-yl)-phenoxymethyl]-quinoline (PF-2545920). This PDE10A inhibitor is the first reported clinical entry fo...
    26: ... Schizophrenia (dagger) dagger Coordinates of the PDE10A crystal structures have been deposited in the Pro...
12. Category:Phosphodiesterase 10a pde10a pde inhibitor (73 bytes)
    1: ...t of pages with the keyword Phosphodiesterase 10a pde10a pde inhibitor
13. 2y0j (3,325 bytes)
    2: ...olines as a novel class of phosphodiesterase 10A (PDE10A) inhibitors, part 2, Lead-optimisation.==
    14: ... novel binding modes to the catalytic site of the PDE10A enzyme.
    16: ...olines as a novel class of phosphodiesterase 10A (PDE10A) inhibitors.,Kehler J, Ritzen A, Langgard M, Pete...
14. 9jdu (2,108 bytes)
    2: ==The crystal structure of PDE10A complexed with inhibitor 2061==
15. 4ael (3,175 bytes)
    2: ==PDE10A in complex with the inhibitor AZ5==
    14: ... was synthesized as potent phosphodiesterase 10A (PDE10A) inhibitors. Structure-based chemical modificatio...
    16: ...naphthyridine-3-carbonitrile derivatives as novel PDE10A inhibitors.,Bauer U, Giordanetto F, Bauer M, O'Ma...
16. 4ddl (3,427 bytes)
    2: ==PDE10a Crystal Structure Complexed with Novel Inhibitor=...
    14: ...d in compound 39, a promising potent inhibitor of PDE10A with good in vivo metabolic stability in rats and...
    16: ...n-3-yl)cinnolines as novel phosphodiesterase 10A (PDE10A) inhibitors.,Hu E, Kunz RK, Rumfelt S, Chen N, Bu...
17. 4dff (3,525 bytes)
    14: ...ound 35 as a potent, selective, and orally active PDE10A inhibitor. Compound 35 inhibited MK-801-induced h...
18. 9ja8 (4,677 bytes)
    14: ...Our findings suggest that effective inhibition of PDE10A potentially confers a protective effect on FMT in...
19. 4lkq (4,054 bytes)
    2: ==Crystal structure of PDE10A2 with fragment ZT017==
    14: ...elding high-resolution co-crystal structures with PDE10A. The structural information was used to elaborate...
    16: Identification and Optimization of PDE10A Inhibitors Using Fragment-Based Screening by Nano...
20. 4llj (4,021 bytes)
    2: ==Crystal structure of PDE10A2 with fragment ZT214==
    14: ...elding high-resolution co-crystal structures with PDE10A. The structural information was used to elaborate...
    16: Identification and Optimization of PDE10A Inhibitors Using Fragment-Based Screening by Nano...

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