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2r9f
From Proteopedia
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[[Image:2r9f.png|left|200px]] | [[Image:2r9f.png|left|200px]] | ||
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{{STRUCTURE_2r9f| PDB=2r9f | SCENE= }} | {{STRUCTURE_2r9f| PDB=2r9f | SCENE= }} | ||
===Calpain 1 proteolytic core inactivated by ZLAK-3002, an alpha-ketoamide=== | ===Calpain 1 proteolytic core inactivated by ZLAK-3002, an alpha-ketoamide=== | ||
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{{ABSTRACT_PUBMED_18702462}} | {{ABSTRACT_PUBMED_18702462}} | ||
==About this Structure== | ==About this Structure== | ||
| - | + | [[2r9f]] is a 1 chain structure with sequence from [http://en.wikipedia.org/wiki/Rattus_norvegicus Rattus norvegicus]. Full crystallographic information is available from [http://oca.weizmann.ac.il/oca-bin/ocashort?id=2R9F OCA]. | |
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| + | ==See Also== | ||
| + | *[[Calpain|Calpain]] | ||
==Reference== | ==Reference== | ||
| - | <ref group="xtra">PMID: | + | <ref group="xtra">PMID:018702462</ref><references group="xtra"/> |
[[Category: Calpain-1]] | [[Category: Calpain-1]] | ||
[[Category: Rattus norvegicus]] | [[Category: Rattus norvegicus]] | ||
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[[Category: Qian, J.]] | [[Category: Qian, J.]] | ||
[[Category: Alpha-ketoamide]] | [[Category: Alpha-ketoamide]] | ||
| - | [[Category: Calcium]] | ||
| - | [[Category: Cytoplasm]] | ||
[[Category: Hydrolase]] | [[Category: Hydrolase]] | ||
[[Category: Inhibitor]] | [[Category: Inhibitor]] | ||
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[[Category: Protease]] | [[Category: Protease]] | ||
[[Category: Thiol protease]] | [[Category: Thiol protease]] | ||
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| - | ''Page seeded by [http://oca.weizmann.ac.il/oca OCA ] on Tue Feb 17 05:52:26 2009'' | ||
Revision as of 12:23, 20 October 2012
Contents |
Calpain 1 proteolytic core inactivated by ZLAK-3002, an alpha-ketoamide
Template:ABSTRACT PUBMED 18702462
About this Structure
2r9f is a 1 chain structure with sequence from Rattus norvegicus. Full crystallographic information is available from OCA.
See Also
Reference
- Qian J, Cuerrier D, Davies PL, Li Z, Powers JC, Campbell RL. Cocrystal structures of primed side-extending alpha-ketoamide inhibitors reveal novel calpain-inhibitor aromatic interactions. J Med Chem. 2008 Sep 11;51(17):5264-70. Epub 2008 Aug 15. PMID:18702462 doi:10.1021/jm800045t
